Linaclotide
Keywords
- Linaclotide Base
- vakawanda inokwanisika mutengo
- CAS # 851199-59-2
Quick Details
- ProName: Linaclotide
- CasNo: 851199-59-2
- Molecular Formula: C59H79N15O21S6
- Chitarisiko: chena upfu
- Application: kushandiswa okurapa kupatirwa
- DeliveryTime: chiriporipocho ainge atumirwa
- Nhuri: maererano mutengi wacho zvaanoda
- Port: Shenzhen
- ProductionCapacity: 1 Kilogram / Month
- Chakachena: 98%
- Storage: 2 ~ 8 ℃. kudzivirirwa kubva chiedza
- Chifambiso: nendege
- LimitNum: 1 giremu
ukuru
Details
Product: Linaclotide
fanano: Linaclotide Acetate
CAS No.: 851199-59-2
Molecular Formula: C59H79N15O21S6
Molecular Weight: 1526,8
Chitarisiko: White upfu
Chakachena:> 98%
urongwa: NH2-Cys-Cys-Glu-Tyr-Cys-Cys-Asn -Pro-ala-Cys-Thr-Gly-Cys-Tyr-OH
Linaclotide chinhu chakaita zvokugadzirwa, gumi nemana amino iine acid peptide uye agonist pamusoro intestinal guanylate cyclase mhando C (GC-C), izvo zvayakaita akarondedzera guanylin peptide mhuri, pamwe secretagogue, unonyaradza marwadzo uye laxative mabasa. Pamusoro zvokuudzwa nomuromo Kutarisirwa, linaclotide runokusunganidzai uye zvaanopa simba GC-C receptors iri luminal penyika intestinal epithelium. Izvi zvinowedzera wevasungwa pamusoro intracellular cyclic guanosine monophosphate (cGMP), iro rinobva guanosine triphosphate (GTP). cGMP zvaanopa simba ari cystic fibrosis transmembrane conductance regulator (CFTR) uye zvinoita secretion kuti chloride uye bicarbonate munzvimbo intestinal lumen. Izvi kunosimudzira yavaibvisa excretion kupinda lumen uye kunoguma yakawedzera intestinal mvura mvura secretion. Izvi pakupedzisira Inowedzera GI dzaifanoiswa pamusoro intestinal mukati, kunonatsiridza bowel kufamba uye anobatsira kupatira. Inosimudzira extracellular cGMP zvese zvinogona vanoshandisa antinociceptive zvazviri, kuburikidza kwakaita asi kwete zvakazara elucidated mashandiro, kuti kungasanganisira vachisiyanisa inzwi pakati nociceptors zvakawanikwa colonic afferent marwadzo fibers. Linaclotide iri zvishoma woga kubva GI turakiti.