Linaclotide
Hua'ōlelo
- Linaclotide Base
- loa affordable uku
- CAS # 851199-59-2
ka poe ola, Details
- ProName: Linaclotide
- CasNo: 851199-59-2
- Hakakino haʻilula: C59H79N15O21S6
- Helehelena: keʻokeʻo he lepo lā
- Noi: hoʻohana 'ia no ka hoola iho la constipation
- DeliveryTime: ke ake ukana
- Makua: e like me ka Customer ka olelo
- Port: Shenzhen
- ProductionCapacity: 1 Kilogram / mahina
- Maemae: 98%
- Waho pūnaewele: 2 ~ 8 ℃. hoomaluia mai ka malamalama
- Ka halihali: ma ka lewa
- LimitNum: 1 Gram
Kiekie
Nā kikoʻī
Product: Linaclotide
hua'ōlelo'ālike: Linaclotide'ākeka
CAS No.: 851199-59-2
hakakino haʻilula: C59H79N15O21S6
hakakino Weight: 1526,8
helehelena: White i one
maemae:> 98%
kaʻina: NH2-Cys-Cys-Glu-Tyr-Cys-Cys-Asn -Pro-Ala-Cys-Thr-Gly-Cys-Tyr-OH
Linaclotide mea he kemikala, heʻumikumamāhā'aminoʻakikaʻakika'amino a me agonist o intestinal guanylate cyclase type C (GC-C), i mea structurally nā i ka guanylinʻakika'amino ohana, me ka secretagogue, analgesic a me laxative hana. Ma ka moʻolelo hoʻoponopono, linaclotide e hoopaa ana i ka a me ka haʻalele no GC-C receptors aia ma luna o ka luminal ili honua o ka intestinal epithelium. Kēia maoli ka lehulehu o intracellular cyclic guanosine monophosphate (cGMP), i ua loko mai guanosine triphosphate (GTP). cGMP haʻalele no ka cystic fibrosis transmembrane conductance mea hoʻokonukonu (CFTR) a stimulates ka secretion o koloriside a me bicarbonate i loko o ka intestinal lumen. Ua paipai 'ia ka paʻakai excretion i loko o ka lumen a me nā hualoaʻa ma ka māhuahua intestinal loli secretion. He ultimately hōʻeleu GI maalo o intestinal Contents, iaono? Ienoai na naau oʻu ka hele a relieves constipation. Hoomahuahua ae la lakou extracellular cGMP pae i kekahi kulia ka antinociceptive hookoia no, ma ka like ana o keia manawa aole i hiki maopopo elucidatedʻano papa hana, i hiki pū modulation o nociceptors loaʻa ma colonic afferent eha olona. Linaclotide ua minimally ke kemu, mai ka GI'āpana.