Degarelix acetate
Keywords
- Degarelix
- vakawanda inokwanisika mutengo
- CAS # 214766-78-6
Quick Details
- ProName: Degarelix acetate
- CasNo: 214766-78-6
- Molecular Formula: C82H103ClN18O16
- Chitarisiko: chena upfu
- Kushandisa: Enguva Application: Advanced hormo ...
- DeliveryTime: chiriporipocho ainge atumirwa
- Nhuri: maererano mutengi wacho zvaanoda
- Port: Shenzhen
- ProductionCapacity: 2 Kilogram / Month
- Chakachena: 98%
- Storage: 2 ~ 8 ℃. kudzivirirwa kubva chiedza
- Chifambiso: nendege
- LimitNum: 1 giremu
ukuru
Details
Molecular Formula:
C82H103ClN18O16
Hama Molecular Misa:
1632,28 g / mol
CAS-Number:
214766-78-6 (mambure)
Long-rokuti Storage:
-20 ± 15 ° C
fanano:
FE200486
Zvinoteverana:
Ac-D-2-nechomukati-D- 4-CPA-D-3-DEVI-water-4-amino-Phe (L-hydroorotyl) -4-ureido-
D-Phe-Leu-Lys (isopropyl) -Pro-D-ala-NH2 acetate munyu
Minda Application:
Advanced kemikari-zvaanoda prostate carcinoma
Active zvakanyanya zvinhu:
Degarelix Acetate ane LHRH (GnRH) Kanotokonya antagonist, kwakaratidza kuti varwere yemhando kenza yeprostate. Degarelix reversibly uye dose-dependently anovanza gonadotropin uye pabonde steroid mumatunhu kuburikidza zvichivhiringidza nokusungwa endogenous LHRH kuti receptors ayo.
Degarelix akaratidza kuva kanenge kubudirira sezvinobvira leuprolide mu kuraramisa kwevari testosterone kuti vari yakaenzana kana kudzika pane kuti kuonekwa castration.