Degarelix roba
koko
- Degarelix
- julọ ti ifarada owo
- CAS # 214766-78-6
awọn ọna alaye
- ProName: Degarelixroba
- CasNo: 214766-78-6
- Molikula agbekalẹ: C82H103ClN18O16
- Irisi: funfun lulú
- Ohun elo: Fields of Ohun elo: To ti ni ilọsiwaju hormo ...
- DeliveryTime: tọ sowo
- Package: gẹgẹ bi onibara ká ibeere
- Port: Shenzhen
- ProductionCapacity: 2 kilogram / osù
- Ti nw: 98%
- Ibi: 2 ~ 8 ℃. ni idaabobo lati ina
- Transportation: nipa air
- LimitNum: 1 Giramu
superiority
awọn alaye
Molikula agbekalẹ:
C82H103ClN18O16
Ojulumo molikula Ibi:
1632,28 g / mol
CAS-Number:
214766-78-6 (net)
Gun-igba Ibi:
-20 ± 15 ° C
synonym:
FE200486
ọkọọkan:
A.-D-2-Nal-D- 4-CPA-D-3-Pal-Ser-4-amino-Phe (L-hydroorotyl) -4-ureido-
D-Phe-Leu-Lys (isopropyl) -Pro-D-ala-NH2 roba iyọ
Aaye ti Ohun elo:
To ti ni ilọsiwaju homonu-ti o gbẹkẹle itọ kasinoma
Ti nṣiṣe lọwọ nkan na:
Degarelix roba jẹ ẹya LHRH (GnRH) ibudo antagonist, itọkasi fun awọn alaisan pẹlu to ti ni ilọsiwaju-itọ akàn. Degarelix reversibly ati iwọn-dependently suppresses gonadotropin ati ibalopo sitẹriọdu ipele nipa inhibiting awọn abuda ti idagbasoke laarin LHRH si awọn oniwe-iṣan.
Degarelix hàn to wa ni o kere bi munadoko bi leuprolide ni sustaining ipele ti ọja ti o wa ni deede si tabi kekere ju ti ri pẹlu castration.