I-Degarelix acetate
Amagama angukhiye
- Degarelix
- intengo kakhulu okungabizi
- CAS # 214766-78-6
Yekuchumana Quick
- ProName: Degarelix acetate
- CasNo: 214766-78-6
- Formula Yamamolekhula: C82H103ClN18O16
- Ukubukeka: powder emhlophe
- Isicelo: Imikhakha Isicelo: hormo okujulile ...
- DeliveryTime: mpahla ngokushesha
- Iphakethe: ngokuvumelana nezimfuneko yekhasimende
- Port: Shenzhen
- ProductionCapacity: 2 Kilogram / Inyanga
- Uhlanzekile: 98%
- Isigcini: 2 ~ 8 ℃. bavikelekile ukukhanya
- Izinto zokuhamba: ngendiza
- LimitNum: 1 Gram
Ukuphakama
Yekuchumana
Formula Yamamolekhula:
C82H103ClN18O16
Isihlobo Yamamolekhula IMisa:
1632,28 g / Mol
CAS-Number:
214766-78-6 (net)
Isitoreji yesikhathi eside:
-20 ± 15 ° C
Emagama lafanako:
FE200486
ukulandelana:
Ac-D-2-Nal-D- 4-CPA-D-3-Pal-Ser-4-amino-Phe (L-hydroorotyl) -4-ureido-
D-Phe-Leu-Lys (isopropyl) -Pro-D-Ala-NH2 usawoti acetate
Imikhakha Isicelo:
Advanced-hormone engaphansi wendlala carcinoma
Into esisebenzayo:
Degarelix acetate kuyinto LHRH (GnRH) yokwamukela omelene, wabonisa iziguli eziphambili umdlavuza wendlala. Degarelix reversibly futhi umthamo-dependently suppresses gonadotropin futhi ubulili steroid amazinga ngomnyaka ka-ezivimbela yokubopha LHRH endogenous ukuze receptor yayo.
Degarelix yabonisa ukuthi okungenani njengoba nomphumela njengoba leuprolide ekusekeleni amazinga testosterone ukuthi kukhona okulingana noma ngaphansana elibonakala nge castration.