I-Nonapeptide-1
Nonapeptide-1 ulusu omnye ezingwevu nonapeptide. It kunokusetyenziswa iintlobo ezahlukeneyo mhlophe okanye bayibone iimveliso okulungisa.
Anqanda melanin yokuqaphela ngokuphazamisa kunye sisenzo tyrosinase in melanocytes. Nciphisa hyperpigmentation kwaye yenze iindawo mnyama eziye yayonakaliswe ilanga kunye nezifo ezithile.
Interfer ne melanocyte ekhuthazayo hormone (MSH). MSH kwandisa ngexesha lokukhulelwa, ngenxa yeemeko ezithile zonyango (umzekelo, isifo seswekile, isifo Addison kaThixo), kwaye ngenxa yokuba kakhulu elangeni.
Nonapeptide-1, xa iqela 200 ug / ml, ikwazi ziyibuyisela umva ngokupheleleyo Yindibanisela bala lintsundu zomngundo.
Kwi 100 ingqondo micromolar, nonapeptide-1 kunganqanda 25-35% yomsebenzi tyrosinase in imifuziselo zezilwanyana kwaye ukunciphisa isiqulatho bala lintsundu of melanocytes nge 27-43%
ukuphakama
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